Drugs for Silicosis (from DrugBank, HMDB, Dgidb, PharmGKB, IUPHAR, NovoSeek, BitterDB):
(show all 17)
# |
|
Name |
Status |
Phase |
Clinical Trials |
Cas Number |
PubChem Id |
1 |
|
Rifapentine |
Approved, Investigational |
Phase 3 |
|
61379-65-5 |
6323497 |
Synonyms:
(2R,16S,17R,18R,19R,20S,21S,22S,23S)-8-{[(4-CYCLOPENTYLPIPERAZIN-1-YL)IMINO]METHYL}-5,6,9,17,19-PENTAHYDROXY-23-METHOXY-2,4,12,16,18,20,22-HEPTAMETHYL-1,11-DIOXO-1,2-DIHYDRO-2,7-(EPOXYPENTADECA[1,11,13]TRIENOIMINO)NAPHTHO[2,1-B]FURAN-21-YL ACETATE
(2S,12Z,14E,16S,17S,18R,19R,20R,21S,22R,23S,24E)-8-{(E)-[(4-cyclopentylpiperazin-1-yl)imino]methyl}-5,6,9,17,19-pentahydroxy-23-methoxy-2,4,12,16,18,20,22-heptamethyl-1,11-dioxo-1,2-dihydro-2,7-(epoxypentadeca[1,11,13]trienoimino)naphtho[2,1-b]furan-21-yl acetate
3-(((4-Cyclopentyl-1-piperazinyl)imino)methyl)rifamycin
3-(((4-cyclopentyl-1-piperazinyl)imino)methyl)rifamycin SV
3-(4-Cyclopentyl-1-piperazinyl)iminomethylrifamycin SV
3-(N-(4-Cyclopentyl-1-piperazinyl)formimidoyl)rifamycin
3-[N-(4-Cyclopentyl-1-piperazinyl)formimidoyl]rifamycin
61379-65-5
71950-35-1
Ambap127923-87-9
Antibiotic DL 473IT
BIDD:GT0669
C08059
C47H64N4O12
CHEBI:45304
CHEMBL1660
CID6323497
CID6434610
CID6835847
CID9919168
CPD000466332
CPD001906779
Cyclopentyl rifampin
Cyclopentylrifampicin
D00879
DB01201
DL 473
DL 473-IT
DL473
DL-473
DL-4-73
DRG-0283
EINECS 262-743-9
|
HMS2051D16
KTC 1
LS-143825
M000473
MDL 473
MDL473
MDL-473
MLS000759441
MLS001424209
NCGC00167431-01
Priftin
Priftin (TN)
Priftin, Cyclopentylrifampicin, Rifapentine
R 77-3
R-773
Rifamycin AF/ACPP
Rifapentin
Rifapentina
Rifapentina [Spanish]
Rifapentine
RIFAPENTINE
Rifapentine (USAN/INN)
Rifapentine [USAN:BAN:INN]
Rifapentinum
Rifapentinum [Latin]
RPE
RPT
S1760_Selleck
SAM001246620
SAM002589953
SMR000466332
UNII-XJM390A33U
|
|
2 |
|
Isoniazid |
Approved, Investigational |
Phase 3 |
|
54-85-3 |
3767 |
Synonyms:
37271-10-6
41466-07-3
4-pyridinecarbohydrazide
4-Pyridinecarbohydrazide
5015 R.P
5015 R.P.
5015 RP
54-85-3
62229-51-0
7640-37-1
AB00052025
Abdizide
AC1L1GNZ
AC1Q54UP
AC1Q54UQ
Acid vanillylidenehydrazide, isonicotinic
AI3-23936
AKOS000119062
Andrazide
Anidrasona
Antimicina
Antituberkulosum
Armacide
Armazid
Armazide
Atcotibine
AZT + Isoniazid
Azuren
bacillen
Bacillin
BB_SC-6246
BIDD:GT0140
Biomol-NT_000288
bp 5 015
BP 5015
BPBio1_000025
BPBio1_001322
BSPBio_000021
BSPBio_002204
C07054
C6H7N3O
CAS-54-85-3
CCRIS 351
Cedin
Cedin (Aerosol)
Cemidon
CHEBI:6030
CHEMBL64
Chemiazid
Chemidon
CID3767
Continazine
Cortinazine
Cotinazin
Cotinizin
CPD000059082
D00346
D007538
DB00951
Defonin
Dibutin
Diforin
Dinacrin
Ditubin
DivK1c_000070
Dow-Isoniazid
Ebidene
EINECS 200-214-6
Eralon
Ertuban
Eutizon
Evalon
Fetefu
Fimalene
FRS-3
FSR 3
FSR-3
Ftivazide
GINK
HIA
Hid rasonil
Hidranizil
Hidrasonil
Hidrulta
Hidrun
HMS1568B03
HMS1920H09
HMS2089I16
HMS2091N19
HMS500D12
HSDB 1647
Hycozid
Hydra
Hydrazid
Hydrazide
Hydrazide, isonicotinic acid
Hyozid
Hyzyd
I.A.I
I.A.I.
I0138
I14-9731
I3377_FLUKA
I3377_SIGMA
IDI1_000070
Ido-tebin
Idrazil
In-73
Inah
INH
Inh-Burgthal
INHd20
Inizid
Iscotin
Isidrina
Ismazide
Isobicina
Isocid
Isocidene
isoco tin
Isocotin
Isohydrazide
Isokin
Isolyn
Isonerit
Isonex
Isoniacid
isoniazid
Isoniazid
Isoniazid & EEP
Isoniazid & Propolis
Isoniazid SA
Isoniazida
Isoniazide
Isoniazidum
Isonicazide
Isonicid
Isonico
Isonicotan
Isonicotil
Isonicotinate hydrazide
Isonicotinhydrazid
Isonicotinic acid hydrazide
Isonicotinic acid vanillylidenehydrazide
Isonicotinic hydrazide
Isonicotinohydrazide
Isonicotinoyl hydrazide
Isonicotinoylhydrazide
Isonicotinsaeurehydrazid
Isonicotinsäurehydrazid
Isonicotinyl hydrazide
Isonicotinyl hydrazine
Isonicotinylhydrazine
Isonide
Isonidrin
Isonikazid
Isonilex
Isonin
Isonindon
Isonirit
|
Isoniton
Isonizida
Isonizide
Isopyrin
Isotamine
Isotebe
Isotebezid
Isotinyl
Isozid
isozid e
Isozide
Isozyd
KBio1_000070
KBio2_001333
KBio2_003901
KBio2_006469
KBio3_001424
KBioGR_000423
KBioSS_001333
L 1945
Laniazid
Laniazid (TN)
Laniozid
LANIZID
LS-205
MLS000069444
MLS001055327
MolPort-000-141-557
Mybasan
NCGC00016244-01
NCGC00016244-02
NCGC00022648-03
NCGC00022648-04
NCGC00022648-05
NCGC00022648-06
nchembio884-comp3
Neoteben
Neo-Tizide
Neoxin
Neumandin
Nevin
Niadrin
Nicazide
Nicetal
Nicizina
Niconyl
Nicotibina
Nicotibine
Nicotisan
Nicozide
Nidaton
nidra zid
Nidrazid
Nikozid
NINDS_000070
Niplen
Nitadon
Niteban
Nitebannsc 9659
NSC 9659
NSC9659
Nydrazid
Nyscozid
Oprea1_396155
Pelazid
Percin
Phthisen
Phthivazid
Phthivazide
Preparation 6424
Prestwick_578
Prestwick0_000161
Prestwick1_000161
Prestwick2_000161
Prestwick3_000161
Pycazide
Pyreazid
Pyricidin
Pyridicin
Pyridine-4-carboxylate hydrazide
Pyridine-4-carboxylic acid hydrazide
Pyrizidin
Raumanon
Razide
Retozide
Rifamate
Rimicid
rimif on
Rimifon
Rimiphone
Rimitsid
Robiselin
Robisellin
Roxifen
RP 5015
RP-5015
RU-EF-Tb
RY-EF-Tb
S1937_Selleck
SAM002554904
Sanohidrazina
Sauterazid
Sauterzid
SMR000059082
SPBio_000094
SPBio_001942
Spectrum_000853
SPECTRUM1500355
Spectrum2_000107
Spectrum3_000472
Spectrum4_000022
Spectrum5_000876
Stanozide
STK086288
TB-Phlogin
TB-Razide
TB-Vis
Tebecid
tebemid
Tebenic
Tebexin
Tebilon
Tebos
Teebaconin
Tekazin
Tibazide
Tibemid
Tibiazide
Tibinide
Tibison
Tibivis
Tibizide
Tibusan
Tisin
Tisiodrazida
Tizide
Tubazid
Tubazide
Tubeco
Tubecotubercid
tubercid
Tuberian
Tubicon
Tubilysin
Tubizid
Tubomel
Tyvid
Unicocyde
Unicozyde
UNII-V83O1VOZ8L
Usaf cb-2
Vanillylidenehydrazide, isonicotinic acid
Vazadrine
Vederon
WLN: T6NJ DVMZ
Zidafimia
Zinadon
ZINC00001590
Zonazide
|
|
3 |
|
Antitubercular Agents |
|
Phase 3 |
|
|
|
4 |
|
Anti-Infective Agents |
|
Phase 3 |
|
|
|
5 |
|
Hypolipidemic Agents |
|
Phase 3 |
|
|
|
6 |
|
Anti-Bacterial Agents |
|
Phase 3 |
|
|
|
7 |
|
Lipid Regulating Agents |
|
Phase 3 |
|
|
|
8 |
|
Antibiotics, Antitubercular |
|
Phase 3 |
|
|
|
9 |
|
Antimetabolites |
|
Phase 3 |
|
|
|
10 |
|
Nintedanib |
Approved |
Phase 2 |
|
656247-17-5 |
56843413 |
Synonyms:
BIBF 1120
BIBF1120
methyl (3Z)-3-[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}anilino)(phenyl)methylidene]-2-oxo-2,3-dihydro-1H-indole-6-carboxylate
|
nintedanib
Nintedanib
Vargatef
|
|
11 |
|
Mitogens |
|
Phase 1, Phase 2 |
|
|
|
12 |
|
Cocaine |
Approved, Illicit |
|
|
50-36-2 |
446220 5760 |
Synonyms:
(−)-cocaine
(-)-Cocaine
(-)-Cocaine base
(1R,2R,3S,5S)-2-(methoxycarbonyl)tropan-3-yl benzoate
(1R,2R,3S,5S)-2-Methoxycarbonyltropan-3-yl benzoate
(R)-Cocaine
[1R-(exo,exo)]-3-(Benzoyloxy)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylate, methyl ester
[1R-(exo,exo)]-3-(benzoyloxy)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylic acid, methyl ester
[1R-(exo,exo)]-3-(Benzoyloxy)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylic acid, methyl ester
1-Cocaine
1i7z
1q72
2beta-Carbomethoxy-3beta-benzoxytropane
2-beta-Carbomethoxy-3-beta-benzoxytropane
2-beta-Tropanecarboxylic acid, 3-beta-hydroxy-, methyl ester, benzoate (ester)
2-Methyl-3beta-hydroxy-1alphah,5alphah-tropane-2beta-carboxylate benzoate (ester)
2-Methyl-3beta-hydroxy-1alphah,5alphah-tropane-2beta-carboxylic acid benzoic acid (ester)
2-Methyl-3b-hydroxy-1alphah,5alphah-tropane-2b-carboxylate benzoate (ester)
2-Methyl-3b-hydroxy-1alphah,5alphah-tropane-2b-carboxylic acid benzoic acid (ester)
2-Methyl-3β-hydroxy-1alphah,5alphah-tropane-2β-carboxylate benzoate (ester)
2-Methyl-3β-hydroxy-1alphah,5alphah-tropane-2β-carboxylic acid benzoic acid (ester)
2-methyl-3β-hydroxy-1αH,5αH-tropane-2β-carboxylate benzoate (ester)
3beta-Hydroxy-2beta-tropanecarboxylic acid methyl ester benzoate (ester)
3-Tropanylbenzoate-2-carboxylic acid methyl ester
50-36-2
53-21-4 (hydrochloride)
610089_ALDRICH
610089_FLUKA
AC-16037
AC1L1EK2
AC1L1L2T
AC1L3U2D
AC1L9JBL
AC-20208
Allococaine
Allopseudococaine
Badrock
Bazooka
b-Cocain
Benzoylethylecgonine
Benzoylmethylecgonine
Bernice
Bernice [Street Name]
Bernies
beta-Cocain
Beta-Cocain
Blast
Blizzard
Blow
Blow [Street Name]
Bouncing Powder
Bump
Burese
C" Carrie
C01416
C8912_SIGMA
Cabello
Candy
Carrie
Caviar
Cecil
Cecil [Street Name]
Charlie
CHEBI:27958
Chicken Scratch
Cholly
CID11779748
CID2826
CID446220
CID5760
COC
Coca
Cocain
Cocaina
cocaine
Cocaine
Cocaine (TN)
Cocaine (USP)
Cocaine [BAN]
Cocaine free base
Cocaine Free Base
Cocaine HCL
Cocaine hydrochloride
Cocaine solution
Cocaine-M
cocainum
Cocainum
Cocktail
Coke
Cola
Corine
CPD-9776
Crack
Crack cocaine
D00110
Dama blanca
Dama Blanca
DB00907
DEA No. 9041
Delcaine
Depsococaine
Dextrocaine
DivK1c_000975
|
d-Pseudococaine
D-pseudococaine
Dust
Ecgonine methyl ester benzoate
Ecgonine methyl ester benzoate solution
Ecgonine, methyl ester, benzoate (ester)
EINECS 200-032-7
Eritroxilina
Erytroxylin
Flake
Flake [Street Name]
Flex
Florida Snow
Foo Foo
Freeze
Girl
Girl [Street Name]
Gold dust
Gold Dust
Gold dust [Street Name]
Goofball
Green gold
Green Gold
G-Rock
Happy dust
Happy Dust
Happy dust [Street Name]
Happy powder
Happy Powder
Happy trails
Happy Trails
HCL, Cocaine
Heaven
Hell
HSDB 6469
Hydrochloride, cocaine
IDI1_000975
Isocaine
Isococain
Isococaine
Jam
KBio1_000975
Kibbles n' Bits
Kibbles N' Bits
Kokain
Kokan
Kokayeen
L000836
Lady
Lady [Street Name]
l-Cocain
L-Cocain
L-Cocaine
Leaf
LS-157759
methyl (1S,4R,5R)-3-benzoyloxy-8-methyl-8-azabicyclo[3.2.1]octane-4-carboxylate
methyl (3S,4R)-3-benzoyloxy-8-methyl-8-azabicyclo[3.2.1]octane-4-carboxylate
methyl [1R-(exo,exo)]-3-(benzoyloxy)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylate
Methyl [1R-(exo,exo)]-3-(benzoyloxy)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylate
Methyl [1R-(exo,exo)]-3-(benzoyloxy)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylic acid
Methyl 3-(benzoyloxy)-8-methyl-8-azabicyclo[3.2.1]octane-2-carboxylate
methyl 3-benzoyloxy-8-methyl-8-azabicyclo[3.2.1]octane-4-carboxylate
Methyl 3beta-hydroxy-1alphaH,5alphaH-tropane-2beta-carboxylate benzoate (ester)
Methyl benzoylecgonine
Methyl Benzoylecgonine
MLS002320697
MolPort-002-535-520
MolPort-003-937-722
Moonrocks
NCGC00159467-02
nchembio.284-comp4
Neurocaine
NINDS_000975
Nose candy
Pimp's drug
Pimp's Drug
Prime Time
Pseudoallococaine
Pseudococaine
Rock
Rock [Street Name]
Sleighride
SMR001338843
Snort
Snow
Snow (birds)
Star dust
Star Dust
Star-spangled powder
Star-Spangled Powder
STOCK1N-68258
Sugar
Sweet Stuff
Toke
Toot
Toot [Street Name]
Trails
UNII-I5Y540LHVR
White girl or lady
Yeyo
Zip
β-cocain
|
|
13 |
|
Rifampicin |
Approved |
|
|
13292-46-1 |
5381226 5458213 |
Synonyms:
13292-46-1
1-b]furan-21-yl acetate
3-(((4-Methyl-1-piperazinyl)imino)-methyl)rifamycin
3-(((4-Methyl-1-piperazinyl)imino)methyl)rifamycin SV
3-([(4-Methyl-1-piperazinyl)imino]methyl)rifamycin SV
3-(4-Methylpiperazinyliminomethyl)rifamycin SV
3-(4-Methylpiperazinyliminomethyl)-rifamycin SV
3-[(4-Methyl-1-piperazinyl)iminomethyl]rifamycin SV
3-[[(4-Methyl-1-piperazinyl)imino]-methyl]rifamycin
46713_FLUKA
46713_RIEDEL
62534-43-4
8-(((4-Methyl-1-piperazinyl)imino)methyl)rifamycin SV
8-(4-Methylpiperazinyliminomethyl) rifamycin SV
8-[[(4-Methyl-1-piperazinyl)imino[methyl]rifamycin
8-[[(4-Methyl-1-piperazinyl)imino]methyl]rifamycin sv
8-[[(4-Methylpiperazinyl)imino]methyl]rifamycin sv
83907_FLUKA
83907_SIGMA
8CI)
Abrifam
Archidyn
Arficin
Arzide
AZT + Rifampin
Ba 41166
Ba 41166/E
BA-41166E
Benemicin
Benemycin
BIDD:PXR0014
Bio-0621
BPBio1_000561
BSPBio_000509
C06688
C43H58N4O12
CAS-13292-46-1
CCRIS 551
CHEBI:28077
CHEBI:455936
CHEMBL180
CID5381226
CID5388984
CID5458213
CID5702112
CID6604339
CID6708473
CID6842115
CID6912767
CID6913622
CPD001906767
D00211
DB01045
Dione 21-acetate
Dipicin
DivK1c_000550
Doloresum
DRG-0109
EINECS 236-312-0
Eremfat
Famcin
Fenampicin
HMS1569J11
HMS1920P08
HMS2089F12
HMS2092G09
HMS501L12
HSDB 3181
KBio1_000550
KBio2_000919
KBio2_003487
KBio2_006055
KBio3_003018
KBioGR_001780
KBioSS_000919
L-5103
L-5103 Lepetit
LS-7689
MLS000028552
MLS001148237
MLS001333745
MolPort-000-767-051
MolPort-002-513-586
MolPort-003-666-281
MolPort-006-395-891
NCGC00016699-01
NCGC00017365-01
NCGC00018178-01
NCGC00022678-03
NCGC00022678-04
NCGC00022678-05
NCGC00160500-01
nchembio884-comp4
|
NCI60_000309
NINDS_000550
NSC 113926
NSC113926
NSC-113926
Piperine & Rifampicin
Prestwick_833
Prestwick0_000525
Prestwick1_000525
Prestwick2_000525
Prestwick3_000525
R/AMP
R0079
R3501_SIAL
R3501_SIGMA
R5777_SIGMA
R7382_SIGMA
Ramp
RAMP
R-Cin
Reserpine & Rifampicin
Rf
Rfamipicin
RFP
Rifa
Rifadin
Rifadin (TN)
Rifadin I.V
Rifadin I.V.
Rifadin Iv
Rifadin IV
Rifadin, Rimactane, Rifampicin, Rifampin
Rifadine
Rifagen
Rifaldazin
Rifaldazine
Rifaldin
Rifam
Rifamicin AMP
Rifamor
Rifampicin
Rifampicin & EEP
Rifampicin & Propolis
Rifampicin (JP15/INN)
Rifampicin [INN:BAN:JAN]
Rifampicin SV
Rifampicina
Rifampicina [INN-Spanish]
Rifampicine
Rifampicine [French]
Rifampicinum
Rifampicinum [INN-Latin]
rifampin
Rifampin
Rifampin (USP)
Rifampin [USAN]
Rifamsolin
Rifamycin
Rifamycin Amp
Rifamycin AMP
Rifaprodin
Rifcin
Rifinah
Rifobac
Rifoldin
Rifoldine
Riforal
Rimactan
Rimactane
Rimactane (TN)
Rimactazid
Rimactin
Rimactizid
Rimazid
Rimycin
RMP
Rofact
S1764_Selleck
SAM002264646
Sinerdol
SMR000058322
SMR000653525
SPBio_002430
Spectrum_000439
SPECTRUM1500529
Spectrum3_001837
Spectrum4_001250
Spectrum5_002018
STK080143
TNP00313
Tubocin
UNII-VJT6J7R4TR
WLN: V1 WQ A&1 E&1 E1UN- AT6N DNTJ D1
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14 |
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Respiratory System Agents |
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|
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15 |
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Anesthetics |
|
|
|
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16 |
|
protease inhibitors |
|
|
|
|
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Synonyms:
|
17 |
|
HIV Protease Inhibitors |
|
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Interventional clinical trials:
(show all 13)
# |
Name |
Status |
NCT ID |
Phase |
Drugs |
1 |
Effectiveness and Tolerability of Weekly Rifapentine/Isoniazid for 3 Months for Tuberculosis Preventive Treatment: A Randomized Controlled Study in China |
Unknown status |
NCT02430259 |
Phase 3 |
Weekly INH / RRT given by DOT |
2 |
Phase 1 Study of Autologous Bone Marrow Stromal Cells With Modification by Hepatocyte Growth Factor to Treat Silicosis |
Completed |
NCT01977131 |
Phase 1, Phase 2 |
|
3 |
The Nintedanib in Progressive Pneumoconiosis Study (NiPPS): a Collaborative NSW Treatment Trial |
Not yet recruiting |
NCT04161014 |
Phase 2 |
Nintedanib 150 MG [Ofev] |
4 |
Phase-1 Study of Autologous Bone Marrow Cells Intrabronchial Instillation for Patients Silicosis |
Completed |
NCT01239862 |
Phase 1 |
|
5 |
A Multicenter, Randomized, Single-blind, Parallel-group Study of Combined Large Volume WLL With Clinical Grade Umbilical Cord Mesenchymal Stem Cells(MSC) Transplantation for Treatment of Pneumoconiosis |
Completed |
NCT02668068 |
Phase 1 |
|
6 |
Oxidative Stress Biomarkers to Monitor and Early Detect Health Impairment in Workers Exposed to Silica (Caesar Stone) |
Unknown status |
NCT01338064 |
|
|
7 |
DNA-damage Pathways in Workers Exposed to Silica (Caesar Stone) |
Unknown status |
NCT01329003 |
|
|
8 |
Comprehensive Risk Assessment of People With Silicosis: A Population-based Study |
Completed |
NCT02794701 |
|
|
9 |
The Use of Forced Oscillation Technique in the Analysis of Respiratory System in Never-smoking Patients With Silicosis:Pathophysiological Study and Evaluation of Diagnostic Accuracy |
Completed |
NCT01725971 |
|
|
10 |
Specialized Center of Research in Occupational and Immunologic Lung Disease |
Completed |
NCT00005280 |
|
|
11 |
Screening Strategy for Early Diagnosis of Silicosis in At-Risk Populations in Oklahoma |
Recruiting |
NCT04205708 |
|
|
12 |
Short Course Rifapentine and Isoniazid for the Preventive Treatment of Tuberculosis(SCRIPT-TB) |
Recruiting |
NCT03900858 |
|
Isoniazidï¼›Rifapentine |
13 |
Respiratory Impairment in Mucopolysaccharidosis Patients: Impact of Glycosaminoglycans (GAG) on the Proteases/Antiproteases Balance |
Not yet recruiting |
NCT04112602 |
|
|
Cochrane evidence based reviews: silicosis
|